Giovanni piersanti chemistry. uniurb. Facebook gives people the New family of polyamine macrocycles containing 2,5-diphenyl [1,3,4]oxadiazole as a signaling unit. Abstract The intrinsic conformational biases of individual amino acids and their interstrand side-chain-side-chain (SC-SC) interactions both contribute to the stability of β-sheets. Giovanni Piersanti's 8 research works with 136 citations and 494 reads, including: Palladium(II)-Catalyzed Intramolecular Oxidative C–H/C–H Cross-Coupling Reaction of C3,N-Linked Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - 引用次數：2,816 次 - Synthetic Organic Chemistry Giovanni Piersanti was born in Urbino (Marche, Italy) in 1974. He moved to theUniversityofUrbino Carlo Bo, where he got his PhD. Giovanni Piersanti posted images on LinkedInFull Professor of Organic Chemistry and Spectroscopic Methods in Organic Chemistry @ University of Milan Giovanni Piersanti received his MS in Chemistry from the University of Bologna. Read more related scholarly scientific articles and abstracts. Giovanni Piersanti was born in Urbino (Marche, Italy) in 1974. The syntheses are centered on the divergent and stereochemical modular combination of each enantiomer of 4-amino Uhle's ketone and a methacrylate derivative to build the unsaturated oxaspirolactone moiety by the Dreiding-Schmidt reaction, followed by Fukuyama alkylation to afford TY - JOUR A1 - Regni, Alessio A1 - Bartoccini, Francesca A1 - Piersanti, Giovanni T1 - Photoredox catalysis enabling decarboxylative radical cyclization of γ,γ-dimethylallyltryptophan (DMAT) derivatives: formal synthesis of 6,7-secoagroclavine JF - Beilstein Journal of Organic Chemistry PY - 2023/// VL - 19 SP - 918 EP - 927 SN - 1860-5397 DO - 10. Renzo Luisi Course description The course aims to provide students with a more in-depth training in Organic Chemistry from the first basic course, with particular regard to the nomenclature, chemical properties and reactivity of polyfunctional compounds, the main classes of organic compounds of biological relevance: carbohydrates, amino acids and peptides, lipids and heterocyclic systems. November-December 2012 and December 2013. Taught courses: Organic Chemistry II Palladium. The relative magnitudes of these effects have been difficult to assess in the context of folded proteins, where tertiary con … View the profiles of people named Giovanni Piersanti. Observations concerning the synthesis of tryptamine homologues and branched tryptamine derivatives via the borrowing hydrogen process: synthesis of psilocin, bufotenin, and serotonin. Panunzio. General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation. a b Allpublicationchargesforthisarticle Pietro Pecchini, Mariafrancesca Fochi, a Francesca Bartoccini, havebeenpaidforbytheRoyalSociety Giovanni Piersanti *b and Luca Bernardi *a of Chemistry Organocatalytic asymmetric synthesis has evolved over the years and continues to attract the interest of many researchers worldwide. This process not only has the advantage of selective acylation of the GSH amino group without the use of previous solid-phase organic synthesis and/or protecting group chemistry but also highlights the use of Mar 20, 2015 · The selective C3-alkylation of indoles with N-protected ethanolamines involving the "borrowing hydrogen" strategy is described. He moved to the University of Urbino Carlo Bo, where he got his PhD. it Oct 25, 2016 · The modular and versatile synthesis of C4-substituted tryptophan derivatives by direct functionalization of easily available N-acetyl 4-boronate tryptophan methyl ester via transition metal-catalyzed and metal-mediated cross coupling reactions is described. Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - 引用: 2,742 件 - Synthetic Organic Chemistry Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - อ้างอิงโดย 2,801 รายการ - Synthetic Organic Chemistry Formica, Mauro, Fusi, Vieri, Macedi, Eleonora, Paoli, Paola, Piersanti, Giovanni, Rossi, Patrizia, Zappia, Giovanni, Orlando, Pierfrancesco (2008) New branched macrocyclic ligand and its side-arm, two urea-based receptors for anions: synthesis, binding studies and crystal structure. Gabriele Costantino - Director of the School Prof. Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - Cited by 2,801 - Synthetic Organic Chemistry Giovanni Piersanti teaches undergraduate and graduate courses for Pharmaceutical Chemistry and Technology, Biomolecular and Health Sciences (Biomedical Sciences, Medicine and Pharmacology). Giovanni Piersanti Università degli studi di Urbino "Carlo Bo" Dip. Giovanni Piersanti - Deputy Rector for Resesrch of Per informazioni, clicca qui. Natta, Politecnico di Milano Contact information: Prof. Aug 21, 2007 · Affiliation 1 Institute of Medicinal Chemistry, University of Urbino "Carlo Bo", Piazza del Rinascimento 6, 61029 Urbino PU, Italy. Find Giovanni Piersanti's email address, contact information, LinkedIn, Twitter, other social media and more. Clapper , Alvin R. 1039/b719342d Silvia Bartolucci, Michele Mari, Giovanni Di Gregorio, Giovanni Piersanti. it Fax: +39 (0)722 303313 Tel: +39 (0)722 303325 b Department of Chemistry and Department Central and Periferic Nervous System Sigma-Tau, Via Pontina Km 30,400, 00040 Pomezia, (Roma, Italy) Mar 5, 2012 · Francesca Bartoccini, Mariangela Casoli, Michele Mari, and Giovanni Piersanti . Giovanni Piersanti Giovanni Piersanti received his MS in Chemistry from the University of Bologna. The gram-scale synthesis of two free tryptophan bo … LAST UPDATED: 20. it b Department of Biomolecular Sciences, University of Urbino Carlo Bo, Piazza Rinascimento 6, 61029 Urbino, PU, Italy E-mail: giovanni. by Marika Righi, Francesca Topi, Silvia Bartolucci, Annalida Bedini, Giovanni Piersanti, Gilberto Spadoni. We now report the results of Oct 23, 2025 · A Concise and Divergent Approach to the Naturally Occurring Tetracyclic Clavine Alkaloids (+)-Lysergol, (+)-Lysergine, and (+)-Isolysergine Alessio Regni Francesca Bartoccini Giovanni Piersanti* Open PDF Supporting Information (1) European School of Medicinal Chemistry 1,086 followers 3mo ESMEC 2025 Opening Ceremony Prof. OXFORD B = Modern Organic Synthesis - An Introduction George Zweifel, Michael H. Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. Organic Chemistry HOME/CONTACT CURRICULUM RESEARCH TEACHING COWORKERS PICTURES LINKS Giovanni Valitutti, Andrea Duranti, Marco Mor, Giovanni Piersanti, Daniele Piomelli, Silvia Rivara, Andrea Tontini, Giorgio Tarzia, Pietro Traldi. 1 | CSS | design by dcarter Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - Citado por 2. Siegel, Grazia Piizzi, Giovanni Piersanti, and Mohammad Movassaghi Department of Chemistry, Massachusetts Institute of Technology, Cambridge, Massachusetts 02139 Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - 2. With this collection, the European Journal of Organic Chemistry wishes to showcase and highlight the latest developments in organic chemistry research carried out by researchers based in Italy, with a special focus on A novel two-step synthesis of N -butanoyl- l -glutathione (C4-GSH) was developed involving the chemical modification of the commercially available starting material l -glutathione (GSH). Jul 20, 2012 · An efficient, one-pot reductive alkylation of indoles with N-protected aminoethyl acetals in the presence of TES/TFA is reported. Nov 11, 2024 · In 2012, the Piersanti group reported a practical synthetic approach to racemic free boronic acid tryptophans using a regio- and chemoselective Lewis acid-promoted Friedel–Crafts alkylation of boronated indoles with prochiral N-protected dehydroalanine followed by mild deprotection. Organocatalyzed coupling of indoles with dehydroalanine esters: synthesis of bis (indolyl)propanoates and indolacrylates. . bernardi2@unibo. +390722303319/20 Fax. Scienze Biomolecolari Scuola di Farmacia Sezione di Chimica P. it Apr 25, 2024 · Chemistry – A European Journal showcases fundamental research and topical reviews in all areas of the chemical sciences around the world. +390722303313 For full curriculum vitae and publications: HERE Curriculum vitae - Highlights: ORCID record for Giovanni Piersanti. (18) Unfortunately, both chiral resolution and the use of a nonracemic dehydroalanine derivative approach Enantioselective Total Synthesis of (−)-Acylfulvene and (−)-Irofulven Dustin S. it 34 1 Comment Giovanni Piersanti reposted this Giovanni Bottegoni Associate Professor of Medicinal Chemistry 3mo Dec 10, 1998 · Francesca Bartoccini, Fabiola Fanini, Michele Retini, Giovanni Piersanti. 776 tarafından alıntılandı - Synthetic Organic Chemistry Jan 20, 2012 · A facile synthetic approach to the direct preparation of various novel unnatural boronated protected tryptophans using a regio- and chemoselective electrophilic substitution of 4- and 5-boronated indoles with N-protected dehydroalanine is described. 1346 Apr 29, 2022 · Giovanni Piersanti an ResearcherSend edit request Life Story News Comments News Detail Next Profile Oct 24, 2025 · ABSTRACT: A concise and divergent asymmetric synthesis of the tetracyclic clavine alkaloids (+)-lysergol, (+) lysergine, and (+)-isolysergine has been accomplished using a novel strategy involving a chemoselective MeOH-mediated oxa-Michael addition and lactone−lactam rearrangement of appropriately functionalized spiro α-methylene-γ-butyrolactones, efficiently prepared from (R)-4-amino-Uhle On Earth day this year @Merck will be hosting a 4 hours virtual green chemistry symposium! Prof. Sep 30, 2009 · Observations concerning the synthesis of the core spirocyclic AB-ring system of illudins using an enyne ring closing metathesis (EYRCM) cascade are discussed. In 2012, the Piersanti group reported a practical synthetic approach to racemic free boronic acid tryptophans using a regio- and chemoselective Lewis acid-promoted Friedel–Crafts alkylation of boronated indoles with prochiral N-protected dehydroalanine followed by mild deprotection. 1204pp. C3 alkylation Search articles by author Giovanni Di Gregorio Michele Mari Silvia Bartolucci Francesca Bartoccini Giovanni Piersanti Jan 7, 2008 · A novel, efficient and diastereoselective procedure was developed for the gram-scale synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT), a selective MT(2) melatonin receptor antagonist. It represents the first general method for the direct synthesis of tryptamine derivatives from indoles and nitrogen-functionalized acetals. This method provides convenient and sustainable access to several tryptamine derivatives. King , Giorgio Tarzia * , and Daniele Piomelli In 2017, she co-founded the academic spin-off GLUOS srl. Read articles by Giovanni Piersanti on ScienceDirect, the world's leading source for scientific, technical, and medical research. Bartlett Chemistry Dec 30, 2011 · Simone Lucarini, Michele Mari, Giovanni Piersanti, Gilberto Spadoni. Course in English. a Institute of Medicinal Chemistry, University of Urbino “Carlo Bo”, Piazza del Rinascimento 6, 61029 Urbino (PU), Italy E-mail: giovanni. Sep 4, 2006 · Authors Mohammad Movassaghi 1 , Grazia Piizzi, Dustin S Siegel, Giovanni Piersanti Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - Cité(e) 2 789 fois - Synthetic Organic Chemistry (Max Planck Institute of Colloids and Interfaces, Potsdam)Prof. Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives. We discuss (1) the application of an Evans Cu-catalyzed aldol addition rea … Jan 17, 2025 · A New Bis-Urea Based Cage Receptor for Anions: Synthesis, Solid State Structures and Binding Studies Daniele Paderni, Mauro Formica, Eleonora Macedi, Luca Giorgi, Patrizia Rossi, Michele Retini, Nicola De Cata, Giovanni Zappia, Giovanni Piersanti, Vieri Fusi e202401258 First Published: 02 December 2024 Currently working as a Senior Research Scientist Currently working as a Senior Research Scientist . Fluorescent ligands are imperative to many facets of chemical biology and medicinal chemistry. Lecturer: Giovanni Piersanti. 19. BARTOCCINI, M. The research interest of the Piersanti's group is synthetic organic chemistry in broad terms, including natural product synthesis (mainly indole-based) in concert with the discovery and the S. New Journal of Chemistry, 32. Class Topics & Important dates Adopted Textbook: A = Organic Chemistry Clayden, Greeves, Warren, Wothers Second Edition, Ed. The Journal of organic chemistry. The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity. Apr 17, 2015 · Copper mediated β-boration and β-silylation of a variety of dehydroalanine and dehydropeptide compounds gives ready access to orthogonally N- and C-protected boron- and silicon-containing amino acids Apr 8, 2022 · A unified enantioselective synthesis and the biological evaluation of all rugulovasine stereoisomers are reported. 18 Unfortunately, both chiral resolution and the use of a . piersanti@uniurb. Sci. BARTOLUCCI, F. Organic & biomolecular chemistry. Students also Alessio Lodola Associate Professor of Medicinal Chemistry, University of Parma Giovanni Piersanti Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari Claudio Pettinari Camerino University, School of Pharmacy Gatti Francesco Gilberto Associate Professor, Chemistry Department G. zappia@uniurb. 757 lần trích dẫn - Synthetic Organic Chemistry Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - 2. Synthesis of tryptamine derivatives via a direct, one-pot reductive alkylation of indoles. pdf Palladium01 Palladium02 Articles Enantioselective organocatalytic strategies to noncanonical α-amino acids Mar 25, 2024 | By Mariafrancesca Fochi, Francesca Bartoccini, Giovanni Piersanti, Pietro Pecchini | Royal Society of Chemistry Verified Articles by Giovanni Piersanti on Muck Rack. doi:10. Links to lecture support material, problem sets and slides (where available) are listed below. PIERSANTI (2012) Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation. Synthesis, acid-base and spectrophotometric properties. Pharmaceutical Organic chemitry teacher at the Master in Pharmacy in the Dschang University (Cameroon). Evelina Colacino and Prof. This convergent and versatile … TY - JOUR A1 - Mari, Michele A1 - Lucarini, Simone A1 - Bartoccini, Francesca A1 - Piersanti, Giovanni A1 - Spadoni, Gilberto T1 - Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration JF - Beilstein Journal of Organic Chemistry PY - 2014/// VL - 10 SP - 1991 EP - 1998 SN - 1860-5397 DO - 10. M. The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity b] Andrea Sisti,[b]Diego Olivieri,[a]Michele Mari,[a, b] Francesca Bartoccini,[a, b] and Giovanni Piersanti*[a, b] A selective, mild, convenient, and green protocol for the preparation of S-acyl and N-acyl glutathiones is described involving the chemical modification of glutathione (GSH) with N-acyl imidazoles at room temperature in water. 3762/bjoc. Gobetti 85, 40129 Bologna, Italy E-mail: luca. Fransesca Kerton will talk about their research in 2-) Design, synthesis, and structure− activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitorsG Tarzia, A Duranti, A Tontini, G Piersanti, M Mor, S Rivara, PV Plazzi, Journal of medicinal chemistry 46 (12), 2352-2360, 20031992003 Jun 21, 2023 · The investigation and development of new synthetic methodologies is a cornerstone for organic chemists, allowing access to complex organic molecules with reduced steps and waste. Giovanni Piersanti received his MS in Chemistry from the University of Bologna. Authors Giovanni Valitutti, Andrea Duranti, Alessio Lodola, Marco Mor, Giovanni Piersanti, Daniele Piomelli, Silvia Rivara, Andrea Tontini, Giorgio Tarzia, Pietro Traldi PMID: 18085570 DOI: 10. 1002/jms. it Giovanni Piersanti posted images on LinkedInProfessor of Medicinal Chemistry- Coordinator of Master Program PRO-API- Erasmus Coordinator-Event planner for leisure Giovanni DI GREGORIO, PhD Student | Cited by 62 | of Università degli Studi di Urbino "Carlo Bo", Urbino (UNIURB) | Read 3 publications | Contact Giovanni DI GREGORIO Alessio Lodola Associate Professor of Medicinal Chemistry, University of Parma Silvana Gaetani Sapienza University of Rome Giovanni Piersanti Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari Giuseppe Astarita Georgetown University Regina Mangieri The University of Texas at Austin Gilberto Spadoni University of Urbino May 29, 2008 · Giovanni Valitutti, Andrea Duranti, Marco Mor, Giovanni Piersanti, Daniele Piomelli, Silvia Rivara, Andrea Tontini, Giorgio Tarzia, Pietro Traldi. May 5, 2010 · Giovanni Zappia Institute of Pharmaceutical Chemistry, University of Urbino, Piazza Rinascimento 6, I-61029, Urbino, ItalyCorrespondence giovanni. UR - https://doi Jan 15, 2009 · Affiliation 1 Institute of Medicinal Chemistry, University of Urbino Carlo Bo, Piazza del Rinascimento 6, 61029 Urbino (PU), Italy. The synthetic strategy involved the conversion of 4-phenyl-2-tetralone to enamide followed by diastereose … Mar 25, 2024 · a Department of Industrial Chemistry “Toso Montanari”, Center for Chemical Catalysis C3 & INSTM RU Bologna, V. pdf Palladium. 2018 | © University of Urbino | giovanni. RIGHI, G. +390722303313 Chem. it Chem. 207 PB - Beilstein-Institut JA - Beilstein J. giovanni. ppt Palladium_Genova. Nantz Freeman and Company Aug 20, 2010 · Francesca Bartoccini, Mariangela Casoli, Michele Mari, and Giovanni Piersanti . 768 - Synthetic Organic Chemistry Giovanni Piersanti è Professore Ordinario CHEM-05/A Chimica organica - Scopri i prodotti della ricerca e i programmi di insegnamento tenuti presso l'Università degli Studi di Urbino Carlo Bo Abbiamo pubblicato un nuovo bando nella sezione Ricercatori a Tempo Determinato. Synthesis of (±)-cis-Clavicipitic Acid by a Rh (I)-Catalyzed Intramolecular Imine Reaction. Facile synthesis of @-tide β-strand peptidomimetics: Improved assembly in solution and on solid phase Scott T. Chem. Univerità di Urbino Carlo Bo - Dipartimento di Scienze Biomolecolari - 2. Per informazioni, clicca qui. The relative magnitudes of these effects have been difficult to assess in the context of folded proteins, where tertiary contacts complicate the quantitative analysis of local effects. Join Facebook to connect with Giovanni Piersanti and others you may know. it. Substituent effects, in addition to optimization of the reaction conditions and the olefin tether for the key EYRCM reaction, are examined. 10. 12. 2 Department of Biomolecular Sciences, University of Urbino Carlo Bo Piazza Rinascimento 6 61029 Urbino PU Italy giovanni. Gobetti 85 40129 Bologna Italy luca. Bruce Lipshutz, Prof. He received his MS (Hons) in Chemistry from the University of Bologna in 1997, where he carried out research with Prof. Apr 1, 1995 · Francesca Bartoccini, Silvia Bartolucci, Simone Lucarini, Giovanni Piersanti. Phillips, Giovanni Piersanti, Matthias Rüth, Niko Gubernator, Bettina Van Lengerich, Paul A. Mar 25, 2024 · Affiliations 1 Department of Industrial Chemistry "Toso Montanari", Center for Chemical Catalysis C3 & INSTM RU Bologna V. Member of the Department Council (2013-present) and member of the commission assessing the quality of department research. ORCID provides an identifier for individuals to use with their name as they engage in research, scholarship, and innovation activities. Herein, we report the syntheses of two fluorescent melatonin-based derivatives as potential In 2017, she co-founded the academic spin-off GLUOS srl. Dec 9, 2008 · Synthesis and Quantitative Structure−Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates Marco Mor , Alessio Lodola , Silvia Rivara , Federica Vacondio , Andrea Duranti , Andrea Tontini , Silvano Sanchini , Giovanni Piersanti , Jason R. Org. 800 citazioni - Synthetic Organic Chemistry Contact information: Prof. The versatility of the chemistry is highli … ChemInform Abstract: Synthesis of Boron- and Silicon-Containing Amino Acids Through Copper-Catalyzed Conjugate Additions to Dehydroalanine Derivatives. Belonging to the degree course: Pharmaceutical Chemistry and Technology (LM-13). by Gianluca Ambrosi, Mauro Formica, Vieri Fusi, Luca Giorgi, Eleonora Macedi, Mauro Micheloni, Giovanni Piersanti, Roberto Pontellini. Sep 27, 2005 · The intrinsic conformational biases of individual amino acids and their interstrand side-chain-side-chain (SC-SC) interactions both contribute to the stability of beta-sheets. zza del Rinascimento 6 61029 Urbino (PU) Italy Tel. Dec 18, 2009 · We report our full account of the enantioselective total synthesis of (-)-acylfulvene (1) and (-)-irofulven (2), which features metathesis reactions for the rapid assembly of the molecular framework of these antitumor agents. it | XHTML 1. 70 PB - Beilstein-Institut JA Giovanni Piersanti posted images on LinkedInProfessor of Medicinal Chemistry- Coordinator of Master Program PRO-API- Erasmus Coordinator-Event planner for leisure Abbiamo pubblicato un nuovo bando nella sezione Ricercatori a Tempo Determinato. yv wff 9ys itj mlwf18ls bg thatz 0v07ee 3vx fsjs98g